Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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91
Tocris Bioscience™ OG 488 BAPTA-1 AM
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Cell-permeable, fluorescently labeled Ca2+ indicator.
92
Tocris Bioscience™ Lonafarnib
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Potent farnesyl transferase inhibitor
| CAS | 193275-84-2 |
|---|---|
| Chemical Name or Material | 4-[2-[4-[(11R)-3,10-Dibromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl]-1-piperidinyl]-2-oxoethyl]-1-piperidinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H31Br2ClN4O2 |
| Formula Weight | Observed MW: 638.82 |
| Assay Percent Range | >98% |
93
Tocris Bioscience™ JNJ 55511118
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Selective, high affinity negative modulator of AMPA receptors containing TARP-γ8
| CAS | 2036081-86-2 |
|---|---|
| Chemical Name or Material | 5-[2-Chloro-6-(trifluoromethoxy)phenyl]-1,3-dihydro-2H-benzimidazol-2-one |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C14H8ClF3N2O2 |
| Formula Weight | Observed MW: 328.67 |
| Assay Percent Range | >98% |
94
Tocris Bioscience™ JNJ 39758979 Dihydrochloride
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High affinity and selective histamine H4 antagonist; orally bioavailable
| Purity | 98% |
|---|---|
| Chemical Name or Material | 4-[(3R)-3-Amino-1-pyrrolidinyl]-6-(1-methylethyl)-2-pyridinamine dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C11H19N5.2HCl |
| Formula Weight | 294.22 |
95
Tocris Bioscience™ WZ 4002
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Potent mutant-selective EGFR inhibitor
| Target | EGF Receptor Inhibitors |
|---|---|
| CAS | 1213269-23-8 |
| Purity | 0.98 |
| Chemical Name or Material | N-[3-[[5-Chloro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]oxy]phenyl]-2-propenamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H27ClN6O3 |
96
Tocris Bioscience™ AP 20187
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Chemical inducer of protein dimerization; active in vivo
97
Tocris Bioscience™ PF 5006739
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Potent CK1δ/ε inhibitor
| CAS | 1293395-67-1 |
|---|---|
| Chemical Name or Material | 4-[4-(4-Fluorophenyl)-1-[1-(3-isoxazolylmethyl)-4-piperidinyl]-1H-imidazol-5-yl]-2-pyrimidinamine |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C22H22FN7O |
| Formula Weight | Observed MW: 419.46 |
| Assay Percent Range | >98% |
98
Tocris Bioscience™ UoS 12258
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Positive allosteric modulator of AMPA receptors (pEC50 = 5.2 for potentiation of AMPA-mediated currents in vitro)
| CAS | 875927-64-3 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[(2S)-5-(6-Fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C17H19FN2O2S |
| Formula Weight | 334.41 |
99
Tocris Bioscience™ Nor NOHA monoacetate
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Arginase inhibitor
100
Tocris Bioscience™ GNE 9278
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Positive allosteric modulator of NMDA receptors; acts in transmembrane domain
| Product Type | Positive Allosteric Modulator |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C21H27N5O3S |
| Formula Weight | 429.54 |
101
Tocris Bioscience™ JMS 17-2 hydrochloride
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CX3CR1 antagonist
| Product Type | Antagonist |
|---|---|
| Purity | 98% |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C25H26ClN3O.HCl |
| Formula Weight | 456.41 |
102
Tocris Bioscience™ DIM-C-pPhOH
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Nur77 antagonist
| CAS | 151358-47-3 |
|---|---|
| Chemical Name or Material | 1,1-Bis(3'-indolyl)-1-(p-hydroxyphenyl)methane |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H18N2O |
| Formula Weight | Observed MW: 338.408 |
| Assay Percent Range | >98% |
103
Tocris Bioscience™ SAG dihydrochloride
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Dihydrochloride salt of SAG; Smo receptor agonist
| CAS | 2702366-44-5 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3-Chloro-N-[trans-4-(methylamino)cyclohexyl]-N-[[3-(4-pyridinyl)phenyl]methyl]benzo[b]thiophene-2-carboxamide dihydrochloride |
| Recommended Storage | Store at -20°C |
| Formula Weight | Observed MW: 562.98 |
| Assay Percent Range | >99% |
104
Tocris Bioscience™ SR 16832
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PPAR gamma Receptor Antagonists
| CAS | 2088135-12-8 |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at 4°C |
| Synonym | 2-Chloro-N-(6-methoxy-4-quinolinyl)-5-nitrobenzamide |
| Molecular Formula | C17H12ClN3O4 |
| Formula Weight | 357.75 |
105
Tocris Bioscience™ B02
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RAD51 recombinase inhibitor
| CAS | 1290541-46-6 |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at 4°C |
| Synonym | 3-(Phenylmethyl)-2-[(1E)-2-(3-pyridinyl)ethenyl]-4(3H)-quinazolinone |
| Molecular Formula | C22H17N3O |
| Formula Weight | 339.4 |